indoles相关论文
A palladium-catalyzed 2-alkylation of indoles with α-bromo esters is developed by employing a P,P=O ligand.The method f......
A highly enantioselective palladium-catalyzed intermolecular tandem Heck/Cacchi reaction of unactivated alkenes with ort......
Direct C-H bond arylation of indoles with aryl boronic acids catalyzed by palladium nanoparticles en
The C2 arylated indoles are important building blocks of biologically active molecules which are found in many natural p......
Metal-Free Catalyzed Oxidative Trimerization of Indoles by Using NaNO2 to Construct Quaternary Carbo
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Nickel(Ⅱ)-catalyzed enantioselective Friedel-Crafts alkylation of indoles with β-CF3-β-(3-indolyl)ni
The bis(3-indolyl)methanes(BIMs)are very important compounds whichpossess a broad range of biological and pharmacologica......
Electron donor-acceptor complexes have known wide applications for the construction of useful organic products by photoc......
Microwave-assist Synthesis of Zero-Dimensional Fluorescent Silicon Nanoparticles Featuring Excitatio
Fluorescent silicon nanoparticles (SiNPs),as the most attractive zero-dimensional silicon nano materials,plays a vital r......
在氧气氛围中,以2-芳基吲哚和N-乙酰基烯胺为原料,实现了一锅法快速构建三环吲哚啉稠环骨架化合物.该方法具有原料易得、操作简便......
报道了Rh(Ⅲ)催化的N-甲氧基-1h-吲哚-1-甲酰胺与亚砜型叶立德的选择性C(2)-H活化/环化反应.该方法为二氢嘧啶并吲哚酮衍生物的制......
The recent developments in inert chemical bond activation have emerged as very attractive altematives to the traditi......
Transition metal-catalyzed carbene transfer reaction is one of the most notable advances for C-C bond formation reaction......
HFIP-promoted catalyst-free cascade reactions for the synthesis of biologically relevant 3,3-di(indo
The first HFIP-promoted catalyst-free cascade reactions for the synthesis of biologically relevant 3,3-di (indolyl)indol......
Synthesis and preliminary cytotoxic evaluation of substituted indoles as potential anticancer agents
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Synthesis of Tridentate Ligands Based on Chiral Diamines and Their Application to Enantioselective F
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Efficient synthesis of bis(indolyl)methanes catalyzed by(PhCH2PPh3)+Br3-under solvent-free condition
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Catalytic Thiourea Promoted Electrophilic Thiocyanation of Indoles and Aromatic Amines with NCS/NH4S
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
目的 通过变应性鼻炎(allergic rhinitis,AR)动物模型,观察组胺H4受体拮抗剂JNJ 7777120对AR大鼠的影响.方法 60只Wistar大鼠以随......
An environmentally friendly synthesis method for bis(indolyl)methanes has been developed in the presence of sodium laury......
采用三价镓十二烷基硫酸盐作催化剂,在溶剂水中,以Michael加成反应制备吲哚酮类化合物,并对其进行了FT-IR、1H NMR等表征。取吲哚1......
吲哚胺2,3-二加氧酶(idoleamine 2,3- dioxygenase,IDO)的高表达是导致肿瘤免疫耐受的一个重要机制.诱导IDO的表达具有两种信号传导......
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产甲烷条件下从废水污泥中驯化的细菌对吲哚的降解包括两步羰基化反应, 生成中间产物氧化吲哚和靛红. 本文研究了产甲烷条件下细菌......
目的:观察5-HT3受体拮抗剂盐酸托烷司琼与盐酸恩丹西酮预防神经外科开颅术患者术后恶心呕吐(PONV)的有效性和安全性。方法:选择神......
K2CO3碱性条件下,1,4-二氧六环为溶剂,3-取代吲哚化合物与α-氯代肟发生D-A反应,生成相应的的吲哚稠杂环化合物。反应中,α-氯代肟......
利用金(Ⅰ)配合物催化吲哚与丙炔酸乙酯的Friedel-Crafts反应,探讨了最优化的实验条件,并合成了不同结构的β-取代双吲哚丙炔酸乙酯......
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本文报道了一种生物活性的吲哚(三氟甲基)羟基烷酸酯的绿色合成方法.以廉价、无毒、高效的乙酰丙酮铁为催化剂,在水相中通过吲哚衍生......
以吲哚(1)和马来酰亚胺(2)为原料,先以0.2个当量的BF3·0Et2为催化刺,C1CH2CH2C1为溶刺,在回流条件下反应4h,生成3-吲哚琥珀酰亚胺......
New Greener Alternative for Biocondensation of Aldehydes and Indoles Using Lemon Juice: Formation of
This work presents a new greener alternative for biocondensation of aldehydes and indoles for the synthesis of bis- and ......
Synthesis, Characterization, Crystal Studies of (E)-3-(3-(4-Fluorophenyl)-1-isopropyl-1H-indol-2-yl)
We have synthesized and developed single crystals of the title compound (E)-3-(3-(4-fluorophenyl)-1-isopropyl-1H-indol-2......
BACKGROUND Gut tryptophan(Trp)metabolites are produced by microbiota and/or host metabolism.Some of them have been prove......
An efficient method for the conjugate addition of indoles to a variety of chalcones using BiBr3 in ethanol (190 proof) i......